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pirenzepine receptor
Also Known As:
pirenzepine receptors; receptor, pirenzepine
Networked:
1
relevant articles (
0
outcomes,
0
trials/studies)
Bio-Agent Context: Research Results
Amino Acids, Peptides, and Proteins: 1
Proteins: 484843
Membrane Proteins: 10078
Cell Surface Receptors: 2125
G-Protein-Coupled Receptors: 4701
Muscarinic Receptors: 2434
pirenzepine receptor: 1
Neurotransmitter Receptors: 562
Cholinergic Receptors: 3880
Muscarinic Receptors: 2434
pirenzepine receptor: 1
Related Diseases
1.
Neuroblastoma
03/01/1988 - "
The M1-selective (high affinity for pirenzepine) muscarinic acetylcholine receptor (mAChR) antagonist pirenzepine displaced both N-[3H]methylscopolamine [( 3H]NMS) and [3H]quinuclidinylbenzilate from intact human SK-N-SH neuroblastoma cells with a low affinity (Ki = 869-1,066 nM), a result indicating the predominance of the M2 or M3 (low affinity for pirenzepine) receptor subtype in these cells.
"
Related Drugs and Biologics
1.
Muscarinic Receptors (Muscarinic Acetylcholine Receptor)
2.
Pirenzepine