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Aprotinin (Trasylol)

A single-chain polypeptide derived from bovine tissues consisting of 58 amino-acid residues. It is an inhibitor of proteolytic enzymes including CHYMOTRYPSIN; KALLIKREIN; PLASMIN; and TRYPSIN. It is used in the treatment of HEMORRHAGE associated with raised plasma concentrations of plasmin. It is also used to reduce blood loss and transfusion requirements in patients at high risk of major blood loss during and following open heart surgery with EXTRACORPOREAL CIRCULATION. (Reynolds JEF(Ed): Martindale: The Extra Pharmacopoeia (electronic version). Micromedex, Inc, Englewood, CO, 1995)
Also Known As:
Trasylol; Antilysin; Bovine Pancreatic Trypsin Inhibitor; Contrical; Contrykal; Dilmintal; Iniprol; Kontrikal; Kontrykal; Pulmin; Traskolan; Zymofren; Inactivator, Kallikrein-Trypsin; Kallikrein Trypsin Inactivator; BPTI, Basic Pancreatic Trypsin Inhibitor; Basic Pancreatic Trypsin Inhibitor; Bovine Kunitz Pancreatic Trypsin Inhibitor; Kallikrein-Trypsin Inactivator; Kunitz Pancreatic Trypsin Inhibitor; Trypsin Inhibitor, Basic, Pancreatic; Trypsin Inhibitor, Kunitz, Pancreatic
Networked: 1522 relevant articles (156 outcomes, 228 trials/studies)

Relationship Network

Drug Context: Research Results

Experts

1. Dietrich, Wulf: 8 articles (02/2009 - 08/2004)
2. van der Linden, Jan: 7 articles (01/2022 - 08/2005)
3. Taylor, K M: 7 articles (05/2008 - 08/2000)
4. Levy, Jerrold H: 7 articles (02/2008 - 01/2004)
5. Royston, David: 6 articles (01/2022 - 08/2004)
6. Augoustides, John G T: 6 articles (06/2008 - 07/2005)
7. Landis, R C: 6 articles (05/2008 - 08/2000)
8. Artunc, Ferruh: 5 articles (01/2022 - 01/2018)
9. Lindvall, Gabriella: 5 articles (04/2019 - 08/2005)
10. Reeves, Scott T: 5 articles (05/2012 - 08/2008)

Related Diseases

1. Hemorrhage
2. Postoperative Hemorrhage
3. Reperfusion Injury
4. Pancreatitis
5. Stroke (Strokes)

Related Drugs and Biologics

1. Tranexamic Acid (AMCA)
2. Peptide Hydrolases (Proteases)
3. Aprotinin (Trasylol)
4. Antifibrinolytic Agents (Antifibrinolytics)
5. Aminocaproic Acid (6 Aminocaproic Acid)
6. Serine Proteinase Inhibitors (Serine Protease Inhibitors)
7. Protease Inhibitors (Protease Inhibitor)
8. Kallikreins (Kallikrein)
9. Lysine (L-Lysine)
10. Serine Proteases (Serine Protease)

Related Therapies and Procedures

1. Cardiopulmonary Bypass (Heart-Lung Bypass)
2. Therapeutics
3. Blood Transfusion (Blood Transfusions)
4. Coronary Artery Bypass (Coronary Artery Bypass Surgery)
5. Orthopedic Procedures