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RPR260243

small molecule activator of the human ether-a-go-go-related gene (HERG) cardiac K+ channel; structure in first source
Also Known As:
(3R,4R)-4-(3-(6-methoxyquinolin-4-yl)-3-oxo-propyl)-1-(3-(2,3,5-trifluoro-phenyl)-prop-2-ynyl)-piperidine-3-carboxylic acid
Networked: 4 relevant articles (0 outcomes, 0 trials/studies)

Bio-Agent Context: Research Results

Experts

1. Chang, Cherlene: 1 article (01/2020)
2. Claydon, Thomas W: 1 article (01/2020)
3. Claydon, Victoria E: 1 article (01/2020)
4. Faizi, Shoaib: 1 article (01/2020)
5. Gunawan, Marvin: 1 article (01/2020)
6. Kemp, Jacob: 1 article (01/2020)
7. Lin, Eric: 1 article (01/2020)
8. Pang, ZhaoKai: 1 article (01/2020)
9. Rayani, Kaveh: 1 article (01/2020)
10. Shafaattalab, Sanam: 1 article (01/2020)

Related Diseases

1. Cardiac Arrhythmias (Arrythmia)
2. Channelopathies
3. Long QT Syndrome
4. Heart Diseases (Heart Disease)

Related Drugs and Biologics

1. Voltage-Gated Potassium Channels (Voltage-Gated Potassium Channel)
2. Cations
3. Carboxylic Acids
4. dofetilide (Tikosyn)
5. piperidine