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BRL 52974
Also Known As:
5-((3,4-dichlorophenyl)acetyl)-4-(1-pyrrolidinylmethyl)-4,5,6,7-tetrahydro-1H-imidazo(4,5-c)pyridine; BRL-52974
Networked:
1
relevant articles (
0
outcomes,
0
trials/studies)
Bio-Agent Context: Research Results
Heterocyclic Compounds: 198
1-Ring Heterocyclic Compounds
Pyrrolidines: 115
BRL 52974: 1
Pyridines: 88
BRL 52974: 1
Experts
1.
Dondio, G
: 1 article (02/2000)
2.
Giardina, G
: 1 article (02/2000)
3.
Hay, D W
: 1 article (02/2000)
4.
Kotzer, C J
: 1 article (02/2000)
5.
Petrillo, P
: 1 article (02/2000)
6.
Underwood, D C
: 1 article (02/2000)
Related Diseases
1.
Cough
02/01/2000 - "
Parenteral administration of selective agonists of the delta-opioid receptor (SB 227122), mu-opioid receptor (codeine and hydrocodone), and kappa-opioid receptor (BRL 52974) produced dose-related inhibition of citric acid-induced cough with ED(50) values of 7.3, 5.2, 5.1, and 5.3 mg/kg, respectively.
"
Related Drugs and Biologics
1.
Citric Acid (Citrate)
2.
kappa Opioid Receptors (kappa Opioid Receptor)
3.
delta Opioid Receptors (delta Opioid Receptor)
4.
mu Opioid Receptors (mu Opioid Receptor)
5.
Hydrocodone (Dihydrocodeinone)
6.
Codeine (Codeine Phosphate)
7.
SB 227122