Abstract |
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Authors | Christoph Boss, Catherine Roch-Brisbare, Michel A Steiner, Alexander Treiber, Hendrik Dietrich, Francois Jenck, Markus von Raumer, Thierry Sifferlen, Christine Brotschi, Bibia Heidmann, Jodi T Williams, Hamed Aissaoui, Romain Siegrist, John Gatfield |
Journal | ChemMedChem
(ChemMedChem)
Vol. 9
Issue 11
Pg. 2486-96
(Nov 2014)
ISSN: 1860-7187 [Electronic] Germany |
PMID | 25147058
(Publication Type: Journal Article)
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Copyright | © 2014 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim. |
Chemical References |
- ACT-462206
- Neurotransmitter Agents
- Orexin Receptor Antagonists
- Orexin Receptors
- Pyrrolidines
- Sulfonamides
- Proline
|
Topics |
- Animals
- Blood-Brain Barrier
(metabolism)
- Brain
(metabolism)
- Dogs
- Half-Life
- Humans
- Madin Darby Canine Kidney Cells
- Male
- Neurotransmitter Agents
(chemistry, pharmacokinetics)
- Orexin Receptor Antagonists
- Orexin Receptors
(metabolism)
- Proline
(chemistry)
- Pyrrolidines
(chemistry, pharmacokinetics)
- Rats
- Rats, Wistar
- Stereoisomerism
- Structure-Activity Relationship
- Sulfonamides
(chemistry, pharmacokinetics)
|