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Pentazocine (Talwin)

The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)
Also Known As:
Talwin; Fortral; Lexir; Pentazocine Hydrochloride; Pentazocine Lactate; Hydrochloride, Pentazocine; Lactate, Pentazocine; 2,6-Methano-3-benzazocin-8-ol, 1,2,3,4,5,6-hexahydro-6,11-dimethyl-3-(3-methyl-2-butenyl)-, (2alpha,6alpha,11R*)-
Networked: 615 relevant articles (35 outcomes, 64 trials/studies)

Relationship Network

Drug Context: Research Results

Experts

1. Smith, Sylvia B: 8 articles (01/2021 - 04/2004)
2. Abe, Fumiaki: 6 articles (08/2008 - 02/2005)
3. Nonaka, Akihiko: 6 articles (08/2008 - 02/2005)
4. Suzuki, Satomi: 6 articles (08/2008 - 02/2005)
5. Marrazzo, Agostino: 4 articles (10/2017 - 01/2011)
6. Prezzavento, Orazio: 4 articles (10/2017 - 01/2011)
7. Ganapathy, Vadivel: 4 articles (01/2011 - 04/2004)
8. Wang, Jing: 3 articles (01/2021 - 01/2016)
9. Fillingim, Roger B: 3 articles (03/2013 - 05/2004)
10. Glover, Toni L: 3 articles (03/2013 - 05/2004)

Related Diseases

1. Pain (Aches)
2. Postoperative Pain
3. Neoplasms (Cancer)
4. Chronic Pain
5. Respiratory Insufficiency (Respiratory Failure)

Related Drugs and Biologics

1. Analgesics (Analgesic Drugs)
2. Morphine (MS Contin)
3. Butorphanol (BC 2627)
4. Meperidine (Pethidine)
5. Diclofenac (SR 38)
6. Pentazocine (Talwin)
7. Buprenorphine (Subutex)
8. Opioid Analgesics (Opioids)
9. Meptazinol
10. Tramadol (K315)

Related Therapies and Procedures

1. Analgesia
2. Cesarean Section (Caesarean Section)
3. Therapeutics
4. Spinal Injections
5. Microspheres (Microsphere)