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gedatolisib

inhibits both phosphatidylinositol 3-kinase and mTOR; structure in first source
Also Known As:
1-(4-((4-(dimethylamino)piperidin-1-yl)carbonyl)phenyl)-3-(4-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)phenyl)urea; PF-05212384; PKI 587; PKI-587; PKI587
Networked: 38 relevant articles (6 outcomes, 14 trials/studies)

Relationship Network

Bio-Agent Context: Research Results

Experts

1. Li, Amin: 2 articles (01/2021 - 01/2019)
2. Ma, Dong: 2 articles (01/2021 - 01/2019)
3. Xie, Yinghai: 2 articles (01/2021 - 01/2019)
4. Xing, Yingru: 2 articles (01/2021 - 01/2019)
5. Zhang, Yinci: 2 articles (01/2021 - 01/2019)
6. Gazi, Mohiuddin: 2 articles (10/2019 - 01/2017)
7. Kazi, Julhash U: 2 articles (10/2019 - 01/2017)
8. Marhäll, Alissa: 2 articles (10/2019 - 01/2017)
9. Moharram, Sausan A: 2 articles (10/2019 - 01/2017)
10. Alsina, Maria: 2 articles (12/2017 - 01/2015)

Related Diseases

1. Neoplasms (Cancer)
2. Colorectal Neoplasms (Colorectal Cancer)
3. Precursor T-Cell Lymphoblastic Leukemia-Lymphoma (T-ALL)
4. Precursor Cell Lymphoblastic Leukemia-Lymphoma (Acute Lymphoblastic Leukemia)
5. Breast Neoplasms (Breast Cancer)

Related Drugs and Biologics

1. mirdametinib
2. ATP-Binding Cassette Transporters (ABC Transporters)
3. palbociclib
4. Estrogen Receptors
5. MTOR Inhibitors
6. 2- amino- 8- (4- (2- hydroxyethoxy)cyclohexyl)- 6- (6- methoxypyridin- 3- yl)- 4- methylpyrido(2,3- d)pyrimidin- 7(8H)- one
7. gedatolisib
8. Mitogen-Activated Protein Kinase Kinases (MEKs)
9. Paclitaxel (Taxol)
10. Irinotecan (Camptosar)

Related Therapies and Procedures

1. Therapeutics
2. Drug Therapy (Chemotherapy)
3. Intravenous Infusions