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dactolisib

antineoplastic agent that inhibits both phosphatidylinositol 3-kinase and mTOR
Also Known As:
2-methyl-2-(4-(3-methyl-2-oxo-8-(quinolin-3-yl)-2,3-dihydroimidazo(4,5-c)quinolin-1-yl)phenyl)propanenitrile; 2-methyl-2-(4-(3-methyl-2-oxo-8-quinolin-3-yl-2,3-dihydro-1h-imidazo(4,5-c)quinolin-1-yl)phenyl)propanenitrile; BEZ235; NVP BEZ235; NVP-BEZ235; NVPBEZ235
Networked: 379 relevant articles (63 outcomes, 101 trials/studies)

Relationship Network

Bio-Agent Context: Research Results

Experts

1. Maira, Sauveur-Michel: 14 articles (01/2014 - 07/2008)
2. Li, Amin: 8 articles (03/2022 - 01/2019)
3. Tang, Xiaolong: 7 articles (12/2021 - 01/2019)
4. Cao, Weiya: 6 articles (12/2021 - 01/2019)
5. Liu, Xueke: 6 articles (12/2021 - 01/2019)
6. Ma, Yongfang: 6 articles (12/2021 - 01/2019)
7. Xu, Ruyue: 6 articles (12/2021 - 01/2019)
8. Zhang, Yinci: 6 articles (12/2021 - 01/2019)
9. García-Echeverría, Carlos: 6 articles (02/2010 - 07/2008)
10. Wu, Binquan: 5 articles (12/2021 - 01/2019)

Related Diseases

1. Neoplasms (Cancer)
2. Breast Neoplasms (Breast Cancer)
3. Neuroblastoma
4. Prostatic Neoplasms (Prostate Cancer)
5. Colorectal Neoplasms (Colorectal Cancer)

Related Drugs and Biologics

1. TOR Serine-Threonine Kinases
2. Phosphatidylinositol 3-Kinases (PI 3 Kinase)
3. dactolisib
4. Phosphotransferases (Kinase)
5. Phosphatidylinositol 3-Kinase (1 Phosphatidylinositol 3 Kinase)
6. Everolimus
7. Sirolimus (Rapamycin)
8. NVP-BKM120
9. AZD 6244
10. Proteins (Proteins, Gene)

Related Therapies and Procedures

1. Therapeutics
2. Drug Therapy (Chemotherapy)
3. Radiotherapy
4. Castration
5. Drug Tapering