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tozasertib

a potent and selective small-molecule inhibitor of the Aurora kinases, suppresses tumor growth
Also Known As:
MK-0457; MK0457; N-(4-((4-(4-methylpiperazin-1-yl)-6-((5-methyl-1H-pyrazol-3-yl)amino)pyrimidin-2-yl)sulfanyl)phenyl)cyclopropanecarboxamide; N-(4-((4-(4-methylpiperazin-1-yl)-6-((5-methyl-1H-pyrazol-3-yl)amino)pyrimidin-2-yl)sulfanyl)phenyl)cyclopropanecarboxamide lactate; N-(4-((4-(4-methylpiperazin-1-yl)-6-((5-methyl-1H-pyrazol-3-yl)amino)pyrimidin-2-yl)sulfanyl)phenyl)cyclopropanecarboxamide, (2S)-2-hydroxypropanoate; VE 465; VE-465; VX-680; VX-680 lactate; VX680; VX680 lactate; cyclopropane carboxylic acid N-(4-(4-(4-methylpiperazin-1-yl)-6-(5-methyl-2H-pyrazol-3-ylamino)pyrimidin-2-ylsulfanyl)phenyl)amide; tozasertib lactate
Networked: 89 relevant articles (5 outcomes, 28 trials/studies)

Relationship Network

Bio-Agent Context: Research Results

Experts

1. Liu, Quentin: 6 articles (11/2013 - 03/2008)
2. Long, Zi-Jie: 4 articles (11/2013 - 08/2009)
3. Yan, Min: 4 articles (11/2013 - 03/2008)
4. Ohyashiki, Kazuma: 4 articles (04/2013 - 06/2008)
5. Okabe, Seiichi: 4 articles (04/2013 - 06/2008)
6. Tauchi, Tetsuzo: 4 articles (04/2013 - 06/2008)
7. Xu, Jie: 4 articles (11/2009 - 03/2008)
8. Tiwari, Vinod: 3 articles (05/2022 - 01/2021)
9. Uniyal, Ankit: 3 articles (05/2022 - 01/2021)
10. Chen, Jia-Jie: 3 articles (01/2020 - 05/2011)

Related Diseases

1. Leukemia
2. Precursor Cell Lymphoblastic Leukemia-Lymphoma (Acute Lymphoblastic Leukemia)
3. Philadelphia Chromosome
4. Carcinoma (Carcinomatosis)
5. Glioblastoma (Glioblastoma Multiforme)

Related Drugs and Biologics

1. Aurora Kinases
2. Vorinostat
3. Carboplatin (JM8)
4. tozasertib
5. Imatinib Mesylate (Gleevec)
6. Histones (Histone)
7. 4- (4- (N- benzoylamino)anilino)- 6- methoxy- 7- (3- (1- morpholino)propoxy)quinazoline
8. Phosphotransferases (Kinase)
9. Adenosine Triphosphate (ATP)
10. Histone Deacetylase Inhibitors

Related Therapies and Procedures

1. Therapeutics
2. Radiotherapy
3. Drug Therapy (Chemotherapy)
4. Stem Cell Transplantation