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B 1086
inhibits p21(ras) farnesyltransferase; methyl ester of B-956
Also Known As:
B-1086
Networked:
2
relevant articles (
0
outcomes,
0
trials/studies)
Bio-Agent Context: Research Results
Organic Chemicals: 133
Sulfur Compounds: 278
Sulfur Amino Acids: 221
Methionine: 6648
B 1086: 2
Amino Acids, Peptides, and Proteins: 1
Amino Acids: 30675
Essential Amino Acids: 1152
Methionine: 6648
B 1086: 2
Sulfur Amino Acids: 221
Methionine: 6648
B 1086: 2
Neutral Amino Acids: 200
Methionine: 6648
B 1086: 2
Experts
1.
Aklilu, F
: 1 article (03/2000)
2.
Gladu, J
: 1 article (03/2000)
3.
Goltzman, D
: 1 article (03/2000)
4.
Rabbani, S A
: 1 article (03/2000)
Related Diseases
1.
Neoplasms (Cancer)
10/15/1997 - "
Treatment in vivo of BALB/c/nu/nu mice bearing Ras-3T3 tumors with B-1086 resulted in a significant inhibition in tumor growth.
"
10/15/1997 - "
We used this system to evaluate the effect of a potent inhibitor of Ras processing, B-1086, on cell growth, PTHRP production, plasma calcium, and tumor growth.
"
03/15/2000 - "
administration of B-1086 (50-100 mg/kg/day) into H-500 tumor-bearing male Fischer rats resulted in a dose-dependent reduction in tumor volume, serum calcium, plasma PTHRP, and tumoral PTHRP mRNA expression.
"
Related Drugs and Biologics
1.
Parathyroid Hormone-Related Protein
2.
Calcium
3.
Messenger RNA (mRNA)