|1.||Liu, Chen-Hai: 1 article (03/2013)|
|2.||Zhu, Cheng-Lin: 1 article (03/2013)|
|3.||Hu, San-Yuan: 1 article (03/2013)|
|4.||Xie, Fang: 1 article (03/2013)|
|5.||Zhu, Kai: 1 article (03/2013)|
|6.||Huang, Qiang: 1 article (03/2013)|
|7.||Estrada-Camarena, Erika: 1 article (01/2013)|
|8.||Gallardo-Tenorio, Alfredo: 1 article (01/2013)|
|9.||Aldrete-Audiffred, Jorge: 1 article (01/2013)|
|10.||Paez-Martinez, Nayeli: 1 article (01/2013)|
03/01/2013 - "An initial immunohistochemistry study of the expressions of GABA receptors in cholangiocarcinoma tissues was followed by the culture and treatment of QBC939 cells for 48 h with GABA, GABA + bicuculine (GABAA receptor antagonist), GABA + phaclofen (GABAB receptor antagonist), and GABA + AG490 (Janus Kinase inhibitor). "
08/01/2004 - "Altered GABAB receptor immunoreactivity in the gerbil hippocampus induced by baclofen and phaclofen, not seizure activity."
07/17/1990 - "However, phaclofen failed to modify the anticonvulsant effect of ethanol against NMDA-induced convulsions. "
07/01/2004 - "Effects of the GABA(B) receptor agonist ((+/-)-baclofen), antagonist (phaclofen), and their combination were tested against clonic seizures induced by cocaine (75 mg/kg). "
07/17/1990 - "The interaction of ethanol with GABAB-receptor system and the selectivity of phaclofen for GABA-receptor subtypes were investigated by employing an in vitro model of 36Cl-influx assay in mammalian cultured neurons and also in vivo models of picrotoxin- and NMDA-induced convulsions in rats. "
07/17/1990 - "Interestingly, phaclofen (200 micrograms i.c.v.) reversed the anticonvulsant effect of ethanol, but not that of pentobarbital or diazepam or progabide, against picrotoxin-induced convulsions in rats. "
11/01/2007 - "Baclofen (150 ng/0.08 microl) increased, whereas phaclofen (300 ng/0.1 microl) reduced the allodynia. "
07/01/2006 - "In naive rats, intrathecal (i.t.) administration in the lumbar spinal cord of GABAA and GABAB receptor antagonists, bicuculline (1-5 microg) and phaclofen (0.1-5 microg), respectively, causes a dose-dependent increase in the magnitude of mechanical allodynia. "
05/01/2002 - "Spinal administration of the GABAA receptor antagonist bicuculline or the GABAB receptor antagonist phaclofen produced tactile allodynia and thermal hyperalgesia in normal rats. "
07/01/2006 - "Inhibitory effects of muscimol and baclofen on both the behavioral mechanical allodynia and the hyperexcitability in WDR neuron with SCI compared to controls, were antagonized by pre-treatment of bicuculline (10 microg) and phaclofen (5 microg), respectively. "
07/01/2004 - "Subcutaneous inoculation of the vector into both feet reduced both manifestations of below-level SCI pain; the vector-mediated effect was partially reversed by intrathecal bicuculline or phaclofen at doses that did not affect thresholds in normal or injured uninoculated animals. "
04/01/2010 - "To these aims, we first analyzed the pain behaviors following the spinal administration of GABA antagonists (1 microg bicuculline/rat and 5 microg phaclofen/rat), agonists (1 microg muscimol/rat and 0.5 microg baclofen/rat) or GABA transporter (GAT) inhibitors (20 microg NNC-711/rat and 1 microg SNAP-5114/rat) into naïve or neuropathic animals. "
01/01/1989 - "Pretreatment with phaclofen significantly decreased the effects of ethanol on motor incoordination, locomotor activity and hypothermia. "
01/01/1989 - "The ability of the GABA(B) receptor antagonist, phaclofen to alter behavioral effects of ethanol was evaluated by loss of righting reflex (sleep time), motor incoordination (bar holding), spontaneous locomotion (open field activity) and hypothermia. "
01/05/2013 - "The hypothermia produced by 4000 ppm toluene was prevented by picrotoxin, bicuculline, phaclofen and finasteride but not by flumazenil. "
|1.||gamma-Aminobutyric Acid (GABA)
|3.||GABA Receptors (GABA Receptor)
|5.||alpha- cyano- (3,4- dihydroxy)- N- benzylcinnamide
|10.||GABA-B Receptor Antagonists